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PAPERS PUBLISHED IN 1995

This list is arranged by the name of the first author. Please, note the change in numbering of the references. Any omissions, mistakes and inconsistencies please communicate to the authors of compilation (michal@5z.com). (If you are pointing to any reference, please use its ID# -- the last number in the reference.) You are welcome to use this compilation in your work. Proper way to quote it in your paper is: Lebl M., Leblova Z.: Dynamic database of references in molecular diversity. Internet http://www.5z.com.


Recently added entries are marked in bold

  1. Anonymous. (1995) Combinatorial chemistry: A strategy for the future - MDL information systems. Net. Sci., 1, #10014 (Available on Internet)

  2. Abraham, R., Buxbaum, S., Link, J., Smith, R., Venti, C., & Darsley, M. (1995) Screening and kinetic analysis of recombinant anti-CEA antibody fragments. J. Immunol. Method, 183, 119-125. #2817

  3. Adey, N.B., Mataragnon, A.H., Rider, J.E., Carter, J.M., & Kay, B.K. (1995) Characterization of phage that bind plastic from phage-displayed random peptide libraries. Gene, 156, 27-31. #4814

  4. Aletras, A., Barlos, K., Gatos, D., Koutsogianni, S., & Mamos, P. (1995) Application of Fmoc-Lys(Mtt)-OH in the preparation of MAPs and MAP-libraries. Epitheor. Klin. Farmacol. Farmakokinet. ,Int. Ed., 9, 129-133. #5825

  5. Ames, R.S., Tornetta, M.A., Deen, K., Jones, C.S., Swift, A.M., & Ganguly, S. (1995) Conversion of murine Fabs isolated from a combinatorial phage display library to full length immunoglobulins. J. Immunol. Method, 184, 177-186. #3190

  6. Ames, R.S., Tornetta, M.A., McMillan, L.J., Kaiser, K.F., Holmes, S.D., Appelbaum, E., Cusimano, D.M., Theisen, T.W., Gross, M.S., Jones, C.S., Silverman, C., Porter, T.G., Cook, R.M., Bennett, D., & Chaiken, I.M. (1995) Neutralizing murine monoclonal antibodies to human IL-5 isolated from hybridomas and a filamentous phage Fab display library. Journal of Immunology, 154, 6355-6364. #4698

  7. Anderson, R.C., Jarema, M.A., Shapiro, M.J., Stokes, J.P., & Ziliox, M. (1995) Analytical techniques in combinatorial chemistry: MAS CH correlation in solvent-swollen resin. J. Org. Chem., 60, 2650-2651. #2638

  8. Anderson, R. C., Jarema, M. A., Shapiro, M. J., Stokes, J. P., and Ziliox, M. NMR techniques in combinatorial chemistry. 1995. #12543

  9. Anderson, R.C., Stokes, J.P., & Shapiro, M.J. (1995) Structure determination in combinatorial chemistry: Utilization of magic angle spinning HMQC and TOCSY NMR spectra in the structure determination of Wang-bound lysine. Tetrahedron Lett., 36, 5311-5314. #2827

  10. Andris, J.S., & Capra, J.D. (1995) The molecular structure of human antibodies specific for the human immunodeficiency virus. J. Clin. Immunol., 15, 17-26. #4684

  11. Antonenko, V.V., Kulikov, N.V., Tumelty, D., Sundaram, A. & Jacobs, J.W. (1995) Combinatorial libraries by light-directed, spatially addressable parallel chemical synthesis: Fidelity of the method and application to drug discovery. In H.L.S. Maia (Ed.), Peptides 94, Proc.23.EPS. (pp. 451-452). ESCOM, Leiden. #2844

  12. Appel, J.R., Buencamino, J., Houghten, R.A. & Pinilla, C. (1995) Study of peptide-antibody interactions using a decapeptide positional scanning library. In H.L.S. Maia (Ed.), Peptides 94, Proc.23.EPS. (pp. 815-816). ESCOM, Leiden. #1311

  13. Baldwin, J.J., Burbaum, J.J., Chelsky, D., Dillard, L.W., Henderson, I., Li, G., Ohlmeyer, M.H.J., Randle, T.L., & Reader, J.C. (1995) Combinatorial libraries encoded with electrophoric tags. Eur. J. Med. Chem., 30 (supplement), 349s-358s. #2807

  14. Baldwin, J.J., Burbaum, J.J., Henderson, I., & Ohlmeyer, M.H.J. (1995) Synthesis of a small molecule combinatorial library encoded with molecular tags. J. Amer. Chem. Soc., 117, 5588-5589. #2737

  15. Bastos, M., Maeji, N.J., & Abeles, R.H. (1995) Inhibitors of human heart chymase based on a peptide library. Proc. Natl. Acad. Sci. USA, 92, 6738-6742. #2878

  16. Bauer, B.E. (1995) The MDL SCREEN approach to the problem of managing data from enterprise-wide high throughput screening (HTS). Net. Sci., 1, #4003 (Available on Internet)

  17. Bianchi, E., Folgori, A., Wallace, A., Nocotra, M., Acali, S., Phalipon, A., Barbato, G., Bazzo, R., Cortese, R., Felici, F., & Pessi, A. (1995) A conformationally homogenous combinatorial peptide library. J. Mol. Biol., 247, 154-160. #2812

  18. Blondelle, S.E., Takahashi, E., Dinh, K.T., & Houghten, R.A. (1995) The antimicrobial activity of hexapeptides derived from synthetic combinatorial libraries. J. Appl. Bacteriol., 78, 39-46. #2682

  19. Blondelle, S.E., Takahashi, E., Houghten, R.A. & Perez-Paya, E. (1995) Design of conformationally defined combinatorial libraries. In H.L.S. Maia (Ed.), Peptides 94, Proc.23.EPS. (pp. 85-86). ESCOM, Leiden. #2831

  20. Blondelle, S.E., Perez-Paya, E., Dooley, C.T., Pinilla, C., & Houghten, R.A. (1995) Soluble combinatorial libraries of organic, peptidomimetics and peptide diversities. TRAC-Trend. Anal. Chem., 14, 83-92. #2692

  21. Bock, J.H., & Slightom, J.L. (1995) Fluorescence-based cycle sequencing with primers selected from a nonamer library. BioTechniques, 19, 60-64. #2735

  22. Boden, P., Eden, J.M., Hodgson, J., Horwell, D.C., Pritchard, M.C., Raphy, J., & Suman-Chauhan, N. (1995) The development of a novel series of non-peptide tachykinin NK(3) receptor selective antagonists. Bioorg. Med. Chem. Lett., 5, 1773-1178. #10539

  23. Boehm, T.L., & Showalter, H.D.H. (1995) Expedient method for the solid-phase synthesis of aspartic acid protease inhibitors directed toward the generation of libraries. Chemtracts:Org. Chem., 8, 331-335. #3466

  24. Boojamra, C.G., Burow, K.M., & Ellman, J.A. (1995) An expedient and high-yielding method for the solid-phase synthesis of diverse 1,4-benzodiazepine-2,5-diones. J. Org. Chem., 60, 5742-5743. #3174

  25. Borman, S. (1995) Liquid-phase combinatorial synthesis technique could ease automation. C&EN, 25-28. #3006

  26. Borrego, B., Wienecke, A., & Schwienhorst, A. (1995) Combinatorial libraries by cassette mutagenesis. Nucl. Acid. Res., 23, 1834-1835. #4664

  27. Bottger, V., Stasiak, P.C., Harrison, D.L., Mellerick, D.M., & Lane, E.B. (1995) Epitope mapping of monoclonal antibodies to keratin 19 using keratin fragments, synthetic peptides and phage peptide libraries. Eur. J. Biochem., 231, 475-485. #2307

  28. Bottger, V., Bottger, A., Lane, E.B., & Spruce, B.A. (1995) Comprehensive epitope analysis of monoclonal anti-proenkephalin antibodies using phage display libraries and synthetic peptides: Revelation of antibody fine specificities caused by somatic mutations in the variable region genes. J. Mol. Biol., 247, 932-946. #3040

  29. Boutillon, C., Diesis, E., Rommens, C., Tartar, A. & Gras-Masse, H. (1995) Combinatorial immunogens: How far can we go? In H.L.S. Maia (Ed.), Peptides 94, Proc.23.EPS. (pp. 845-846). ESCOM, Leiden. #3534

  30. Boyd, S.M., Beverley, M., Norskov, L., & Hubbard, R.E. (1995) Characterising the geometric diversity of functional groups in chemical databases. J. Comput. Aid. Molec. Design, 9, 417-424. #4678

  31. Bradbury, A., & Cattaneo, A. (1995) The use of phage display in neurobiology. Trends Neurosci., 18, 243-249. #3139

  32. Bradshaw, C.G., Magnenat, E. & Chollet, A. (1995) Screening for interactions between suitably labelled proteins and an immobilised cyclic peptide library. In H.L.S. Maia (Ed.), Peptides 94, Proc.23.EPS. (pp. 491-492). ESCOM, Leiden. #2852

  33. Bray, A.M., Valerio, R.M., Dipasquale, A.J., Greig, J., & Maeji, N.J. (1995) Multiple synthesis by the multipin method as a methodological tool. J. Peptide Sci., 1, 80-87. #2599

  34. Bray, A.M., Chiefari, D.S., Valerio, R.M., & Maeji, N.J. (1995) Rapid optimization of organic reactions on solid phase using multipin approach: Synthesis of 4-aminoproline analogues by reductive amination. Tetrahedron Lett., 36, 5081-5084. #2804

  35. Briceno, G., Chang, H., Sun, X., Schulz, P.G., & Xiang, X.D. (1995) A class of cobalt oxide magnetoresistance materials discovered with combinatorial synthesis. Science, 270, 273-275. #3553

  36. Brown, B.B., Wagner, D.S., & Geysen, H.M. (1995) A single-bead decode strategy using electrospray ionization mass spectrometry and a new photolabile linker: 3-Amino-3-(2- nitrophenyl)-propionic acid. Mol. Diversity, 1, 4-12. #2821 (Available on Internet)

  37. Bruce, J.E., Anderson, G.A., Chen, R., Cheng, X., Gale, D.C., Hofstadler, S.A., Schwartz, B.L., & Smith, R.D. (1995) Bio-affinity characterization mass spectrometry. Rapid Commun. Mass Spectrom., 9, 644-650. #3147

  38. Bruno, W.J., Knill, E., Balding, D.J., Bruce, D.C., Doggett, N.A., Sawhill, W.W., Stallings, R.L., Whittaker, C.C., & Torney, D.C. (1995) Efficient pooling designs for library screening. Genomics, 26, 21-30. #6068

  39. Brussolo, J.S., & DeWitt, S.H. (1995) Automated sample handlig systems. Net. Sci., 1, #4000 (Available on Internet)

  40. Burbaum, J.J., Ohlmeyer, M.H.J., Reader, J.C., Henderson, I., Dillard, L.W., Li, G., Randle, T.L., Sigal, N.H., Chelsky, D., & Baldwin, J.J. (1995) A paradigm for drug discovery employing encoded combinatorial libraries. Proc. Natl. Acad. Sci. USA, 92, 6027-6031. #2732

  41. Burger, M.T., & Still, W.C. (1995) Synthetic ionophores. Encoded combinatorial libraries of cyclen- based receptors for Cu(2+) and Co(2+). J. Org. Chem., 60, 7382-7383. #3355

  42. Burioni, R., Plaisant, P., Riccio, M.L., Rossolini, G.M., Santangelo, R., Vannini, A., & Satta, G. (1995) Engineering human monoclonal antibody fragments: A recombinant enzyme-linked Fab. Microbiologica, 18, 127-133. #4655

  43. Burritt, J.B., Quinn, M.T., Jutila, M.A., Bond, C.W., & Jesaitis, A.J. (1995) Topological mapping of neutrophil cytochrome b epitopes with phage-display libraries. Journal of Biological Chemistry, 270, 16974-16980. #3142

  44. Campbell, D.A., Bermak, J.C., Burkoth, T.S., & Patel, D.V. (1995) A transition state analogue inhibitor combinatorial library. J. Amer. Chem. Soc., 117, 5381-5382. #2727

  45. Canne, L.E., Walker, S.M., & Kent, S.B.H. (1995) A general method for the synthesis of thioester resin linkers for use in the solid phase synthesis of peptide-a-thioacids. Tetrahedron Lett., 36, 1217-1220. #2357

  46. Carell, T., Wintner, E.A., Sutherland, A.J., Rebek, J.Jr., Dunayevskiy, Y.M., & Vouros, P. (1995) New promise in combinatorial chemistry: Synthesis, characterization, and screening of small-molecule libraries in solution. Chem. Biol., 2, 171-183. #2640

  47. Cargill, J. F., Maiefski, R. R., and Toyonaga, B. E. Automated combinatorial chemistry on solid phase. In: Anonymous. (Eds.) Zymark Corporation, Hopkinton, MA p.221 Proceedingds of the 13th International Symposium of Laboratory Robotics and Automation 1995. #8300

  48. Carrasco, M.R., & Still, W.C. (1995) Engineering of a synthetic receptor to alter peptide binding selectivity. Chem. Biol., 2, 205-212. #3789

  49. Cattani, P., Plaisant, P., Manzara, S., Capodicasa, N., Burioni, R., Rossolini, G.M., & Satta, G. (1995) Cloning and characterization of human recombinant antibody Fab fragments specific for types 1 and 2 Herpes Simplex virus. Microbiologica, 18, 135-142. #4697

  50. Cesareni, G., Castagnoli, L., Dente, L., Iannolo, G., Vetriani, C., Felici, F., Luzzago, A., Monaci, P., Nicosia, A. & Cortese, R. (1995) Construction and utilization of peptide libraries displayed by filamentous bacteriophage. In N.D. Zegers, W.J.A. Boersma & E. Claassen (Eds.), Immunological Recognition of Peptides in Medicine and Biology. (pp. 44-59). CRC Press,Inc., Boca Raton. #4962

  51. Chabala, J.C., Baldwin, J.J., Burbaum, J.J., Chelsky, D., Dillard, L.W., Henderson, I., Li, G., Ohlmeyer, M.H.J., Randle, T.L., Reader, J.C., Rokosz, L., & Sigal, N.H. (1995) Binary encoded small-molecule libraries in drug discovery and optimization. Perspect. Drug Disc. Design, 2, 305-318. #2905

  52. Chabala, J.C. (1995) Solid-phase combinatorial chemistry and novel tagging methods for identifying leads. Curr. Opin. Biotechnol., 6, 632-639. #4916

  53. Chakravarty, S., Mavunkel, B.J., Andy, R., & Kyle, D. (1995) Non-peptidic bradykinin receptor antagonists from a structurally directed non-peptide library. Net. Sci., 1, #10015 (Available on Internet)

  54. Chen, J., Bernstein, H.S., Chen, M., Wang, L., Ishi, M., Turck, C.W., & Coughlin, S.R. (1995) Tethered ligand library for discovery of peptide agonists. Journal of Biological Chemistry, 270, 23398-23401. #3513

  55. Chen, J.K., & Schreiber, S.L. (1995) Combinatorial synthesis and multidimensional NMR spectroscopy: An approach to understanding protein-ligand interactions. Angew. Chem. Int. Ed., 34, 953-969. #3416

  56. Chinnaiyan, A.M., O'Rourke, K., Tewari, M., & Dixit, V.M. (1995) FADD, a novel death domain-containing protein, interacts with the death domain of Fas and initiates apoptosis. Cell, 81, 505-512. #11192

  57. Chorev, M., Dresner-Pollak, R., Eshel, Y., & Rosenblatt, M. (1995) Approach to discovering novel therapeutic agents for osteoporosis based on integrin receptor blockade. Biopolymers, 37, 367-375. #4826

  58. Chu, S.S., & Reich, S.H. (1995) NPIT: A new reagent for quantitatively monitoring reactions of amines in combinatorial synthesis. Bioorg. Med. Chem. Lett., 5, 1053-1058. #3224

  59. Chu, Y.H., Kirby, D.P., & Karger, B.L. (1995) Free solution identification of candidate peptides from combinatorial libraries by affinity capillary electrophoresis/mass spectrometry. J. Amer. Chem. Soc., 117, 5419-5420. #2738

  60. Cianfriglia, M., Romagnoli, G., Tombesi, M., Poloni, F., Falasca, G., Di Modugno, F., Castagna, M., & Chersi, A. (1995) P-Glycoprotein epitope mapping. II.The murine monoclonal antibody MM6.15 to human multidrug-resistant cells binds with three distinct loops in the MDR1-P-glycoprotein extracellular domain. Int. J. Cancer, 61, 142-147. #4732

  61. Conrad, R.C., Baskerville, S., & Ellington, A.D. (1995) In vitro selection methodologies to probe RNA function and structure. Mol. Diversity, 1, 69-78. #3129 (Available on Internet)

  62. Coombs, G.S., Hazzard, J., & Corey, D.R. (1995) Kinetic characterization of a peptide inhibitor of trypsin isolated from a synthetic peptide combinatorial library. Bioorg. Med. Chem., 5, 611-614. #3417

  63. Cortese, R., Monaci, P., Nicosia, A., Luzzago, A., Felici, F., Galfre, G., Pessi, A., Tramontano, A., & Sollazzo, M. (1995) Identification of biologically active peptides using random libraries displayed on phage. Curr. Opin. Biotechnol., 6, 73-80. #2933

  64. Courtney, B.C., Williams, K.C., & Schlager, J.J. (1995) A phage display vector with improved stability, applicability and ease of manipulation. Gene, 165, 139-140. #4681

  65. Courtney, B.C., Williams, K.C., Bing, Q.A., & Schlager, J.J. (1995) Capillary gel electrophoresis as a method to determine ligation efficiency. Anal. Biochem., 228, 281-286. #6234

  66. Crameri, A., & Stemmer, W.P.C. (1995) Combinatorial multiple cassette mutagenesis creates all the permutations of mutant and wild-type sequences. BioTechniques, 18, 194-196. #2699

  67. Crosby, W.L., & Schorr, P. (1995) Principles and applications of recombinant antibody phage display technology to plant biology. Methods Cell Biol., 50, 85-99. #4151

  68. Cuervo, J.H., Weitl, F., Ostresh, J.M., Hamashin, V.T., Hannah, A.L. & Houghten, R.A. (1995) Polyalkylamine chemical combinatorial libraries. In H.L.S. Maia (Ed.), Peptides 94, Proc.23.EPS. (pp. 465-466). ESCOM, Leiden. #2846

  69. Czarnik, A.W. (1995) Why combinatorial chemistry, why now (and why you should care). Chemtracts:Org. Chem., 8, 13-18. #2809

  70. Dankwardt, S.M., Newman, S.R., & Krstenansky, J.L. (1995) Solid phase synthesis of aryl and benzylpiperazines and their application in combinatorial chemistry. Tetrahedron Lett., 36, 4923-4926. #2805

  71. Dapremont, L., Valerio, R.M., Bray, A.M., Stewart, K.M., Mason, T.J., Wang, A.W., & Maeji, N.J. (1995) Multiple synthesis using the multipin method. Physiol. Chem. Phys. Med. NMR, 27, 339-343. #5215

  72. Davies, K., & White, C. (1995) An information management architecture for combinatorial chemistry. Net. Sci., 1, #5501 (Available on Internet)

  73. Davis, P.W., Vickers, T.A., Wilson-Lingardo, L., Wyatt, J.R., Guinosso, C.J., Sanghvi, Y.S., DeBaets, E.A., Acevedo, O.L., Cook, P.D., & Ecker, D.J. (1995) Drug leads from combinatorial phosphodiester libraries. J. Med. Chem., 38, 4363-4366. #3379

  74. de Koster, H.S., Amons, R., Benckhuijsen, W.E., Feijlbrief, M., Schellekens, G.A., Welling-Wester, S., Welling, G.W. & Drijfhout, J.W. (1995) Complementary synthetic peptide libraries of limited complexity reveal high affinity binding mimotopes. In H.L.S. Maia (Ed.), Peptides 94, Proc.23.EPS. (pp. 851-852). ESCOM, Leiden. #2854

  75. de Koster, H.S., Amons, R., Benckhuijsen, W.E., Feijlbrief, M., Schellekens, G.A., & Drijfhout, J.W. (1995) The use of dedicated peptide libraries permits the discovery of high affinity binding peptides. J. Immunol. Method, 187, 179-188. #4317

  76. de Kruif, J., Boel, E., & Logtenberg, T. (1995) Selection and application of human single chain Fv antibody fragments from a semi-synthetic phage antibody display library with designed CDR3 regions. J. Mol. Biol., 248, 97-105. #3042

  77. de Kruif, J., Terstappen, L., Boel, E., & Logtenberg, T. (1995) Rapid selection of cell subpopulation-specific human monoclonal antibobies from a synthetic phage antibody library. Proc. Natl. Acad. Sci. USA, 92, 3938-3942. #2739

  78. Dean, P.M. (1995) Synthetic peptide combinatorial libraries (SPCLs). Exp. Opin. Ther. Patents, 5, 887-899. #4907

  79. DeLeo, F.R., Yu, L., Burritt, J.B., Loetterle, L.R., Bond, C.W., Jesaitis, A.J., & Quinn, M.T. (1995) Mapping sites of interaction of p47-phox and flavocytochrome b with random-sequence peptide phage display libraries. Proc. Natl. Acad. Sci. USA, 92, 7110-7114. #3138

  80. Deleuze, H., & Sherrington, D.C. (1995) Poly(p-acetoxylstyrene) resin: A prospective new support for combinatorial synthesis. J. Chem. Soc. Perkin Trans. 2, 36, 2217-2221. #5628

  81. Deprez, B., Williard, X., Bourel, L., Coste, H., Hyafil, F. & Tartar, A. (1995) Self-deciphering, orthogonal combinatorial libraries of soluble organic compounds: Discovery of a potent V2 vasopressin antagonist. In H.L.S. Maia (Ed.), Peptides 94, Proc.23.EPS. (pp. 455-456). ESCOM, Leiden. #1673

  82. Deprez, B., Williard, X., Bourel, L., Coste, H., Hyafil, F., & Tartar, A. (1995) Orthogonal combinatorial chemical libraries. J. Amer. Chem. Soc., 117, 5405-5406. #2724

  83. deStevens, G. (1995) Heterocyclic diversity: The road to biological activity. In E. Jucker (Ed.), Progress in Drug Research. (pp. 9-47). Birkh user Verlag, Basel. #3257

  84. DeWitt, S.H., Schroeder, M.C., & Stankovic, C.J. (1995) Integration and automation of multiple, simultaneous organic synthesis on a solid support. Amer. Lab., 26AA-26BB. #2421

  85. DeWitt, S.H. (1995) Combinatorial libraries and high throughput synthesis. In C.G. Wermuth (Ed.), The Practice of Medicinal Chemistry. Academic Press, London. #2419

  86. DeWitt, S.H., & Czarnik, A.W. (1995) Automated synthesis and combinatorial chemistry. Curr. Opin. Biotechnol., 6, 640-645. #8207

  87. Ding, Y., Kanie, O., Labbe, J., Palcic, M.M., Ernst, B. & Hindsgaul, O. (1995) Synthesis and biological activity of oligosaccharide libraries. In A. Alavi & J.S. Axford (Eds.), Advances in Experimental medicine and Biology: Glycoimmunology. (pp. 261-269). Plenum Press, New York. #3811

  88. Ditzel, H.J., Binley, J.M., Moore, J.P., Sodroski, J., Sullivan, N., Sawyer, L.S.W., Hendry, R.M., Yang, W.P., Barbas, C.F.I., & Burton, D.R. (1995) Neutralizing recombinant human antibodies to a conformational V2- and CD4-binding site-sensitive epitope of HIV-1 gp120 isolated by using an epitope-masking procedure. Journal of Immunology, 154, 893-906. #2272

  89. Domingo, G.J., Leatherbarrow, R.J., Freeman, N., Patel, S., & Weir, M. (1995) Synthesis of a mixture of cyclic peptides based on the Bowman-Birk reactive site loop to screen for serine protease inhibitors. Int. J. Peptide Prot. Res., 46, 79-87. #2729

  90. Dooley, C.T., & Houghten, R.A. (1995) Identification of mu-selective polyamine antagonists from a synthetic combinatorial library. Analgesia, 1, 400-404. #9383

  91. Dooley, C.T., Kaplan, R.A., Chung, N.N., Schiller, P.W., Bidlack, J.M., & Houghten, R.A. (1995) Six highly active Mu-selective opioid peptides identified from two synthetic combinatorial libraries. Peptide Res., 8, 124-137. #2726

  92. Dooley, C.T., & Houghten, R.A. (1995) A comparison of combinatorial library approaches for the study of opioid compounds. Perspect. Drug Disc. Design, 2, 287-304. #2904

  93. Dooley, C.T., Hope, S.K. & Houghten, R.A. (1995) Identification of tetrameric opioid peptides from a combinatorial library composed of L-, D- and non-proteinogenic amino acids. In H.L.S. Maia (Ed.), Peptides 94, Proc.23.EPS. (pp. 805-806). ESCOM, Leiden. #1837

  94. Dorner, B., Ostresh, J.M., Husar, G.M. & Houghten, R.A. (1995) Extending the range of molecular diversity through amide alkylation of peptide libraries. In H.L.S. Maia (Ed.), Peptides 94, Proc.23.EPS. (pp. 463-464). ESCOM, Leiden. #1606

  95. Duenas, M., Ayala, M., Vazquez, J., Ohlin, M., Soderlind, E., Borrebaeck, C.A.K., & Gavilondo, J.V. (1995) A point mutation in a murine immunoglobulin V-region strongly influences the antibody yield in Escherichia coli. Gene, 158, 61-66. #2819

  96. Dunayevskiy, Y.M., Vouros, P., Carell, T., Wintner, E.A., & Rebek, J.Jr. (1995) Characterization of the complexity of small molecule libraries by electrospray ionization mass spectrometry. Anal. Chem., 67, 2906-2915. #3192

  97. Dybwad, A., Forre, O., Natvig, J.B., & Sioud, M. (1995) Structural characterization of peptides that bind synovial fluid antibodies from RA patients: A novel strategy for identification of disease-related epitopes using a random peptide library. Clin. Immunol. Immunopathol., 75, 45-50. #4731

  98. Ecker, D.J., & Crooke, S.T. (1995) Combinatorial drug discovery: Which methods will produce the greatest value? Biotechnology, 13, 351-360. #4056

  99. Eden, J., Hodgson, J., Horwell, D.C., Howson, W., Pritchard, M.C. & Raphy, J. (1995) The development of a high affinity NK(3) receptor antagonist. In H.L.S. Maia (Ed.), Peptides 94, Proc.23.EPS. (pp. 712-713). ESCOM, Leiden. #2853

  100. Efimov, V.P., Nepluev, I.V., & Mesyanzhinov, V.V. (1995) Bacteriophage T4 as a surface display vector. Virus Genes, 10, 173-177. #3252

  101. Egner, B.J., Langley, G.J., & Bradley, M. (1995) Solid phase chemistry: Direct monitoring by matrix-assisted laser desorption/ionization time of flight mass spectrometry.A tool for combinatorial chemistry. J. Org. Chem., 60, 2652-2653. #2639

  102. Eichler, J., Lucka, A.W. & Houghten, R.A. (1995) Cyclic peptide template synthetic combinatorial libraries. In H.L.S. Maia (Ed.), Peptides 94, Proc.23.EPS. (pp. 461-462). ESCOM, Leiden. #1684

  103. Eichler, J., Appel, J.R., Blondelle, S.E., Dooley, C.T., Dorner, B., Ostresh, J.M., Perez-Paya, E., Pinilla, C., & Houghten, R.A. (1995) Peptide, peptidomimetic, and organic synthetic combinatorial libraries. Med. Res. Rev., 15, 481-496. #3470

  104. Eichler, J., & Houghten, R.A. (1995) Generation and utilization of synthetic combinatorial libraries. Mol. Med. Today, 1, 174-180. #3199

  105. Ellman, J.A. (1995) Combinatorial organic libraries. Chemtracts:Org. Chem., 8, 1-4. #2161

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