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PAPERS PUBLISHED IN 2002

This list is arranged by the name of the first author. Any omissions, mistakes and inconsistencies please communicate to the authors of compilation (michal@5z.com). (If you are pointing to any reference, please use its ID# -- the last number in the reference.) You are welcome to use this compilation in your work. Proper way to quote it in your paper is: Lebl M., Leblova Z.: Dynamic database of references in molecular diversity. Internet http://www.5z.com.

Recently added entries are marked in bold

  1. Agrafiotis,D.K. (2002) Multiobjective optimization of combinatorial libraries. J. Comput. Aid. Molec. Design, 16, 335-356. #17479

  2. Agrafiotis,D.K., Lobanov,V.S., & Salemme,F.R. (2002) Combinatorial informatics in the post-genomics era. Nature Reviews Drug Discovery, 1, 337-346. #17648

  3. Ahmet,P., Koida,T., Takakura,M., Nakajima,K., Yoshimoto,M., Koinuma,H., Tanaka,M., Takeguchi,M., & Chikyow,T. (2002) Diffusion induced amorphization in the crystalline SrTiO3 thin films grown on Si (100) investigated by combinatorial method. Applied Surface Science, 189, 307-312. #17617

  4. Ajay. (2002) Predicting drug-likeness: why and how? Current Topics in Medicinal Chemistry (Hilversum, Netherlands), 2, 1273-1286. #17466

  5. Amis,E.J., Xiang,X.D., & Zhao,J.C. (2002) Combinatorial materials science: What's new since Edison? MRS Bulletin, 27, 295-300. #17693

  6. Andrec,M., & Levy,R.M. (2002) Protein sequential resonance assignments by combinatorial enumeration using 13C.alpha. chemical shifts and their (i, i-1) sequential connectivities. J. Biomol. NMR, 23, 263-270. #17516

  7. Anon. (2002) 2nd eurasian meeting on heterocyclic chemistry \"heterocycles in organic and combinatorial chemistry\". Asian Journal of Chemistry, 14, 1229. #17540

  8. Anon. (2002) Combinatorial chemistry: Torial set to speed catalysts to market. Chemistry & Industry (London, United Kingdom), 6. #17545

  9. Anon. (2002) Recent patents in combinatorial chemistry. Nat. Biotech., 20, 745. #17599

  10. Anon. (2002) Two Medicinal Fellows to give presentations. Chemical & Engineering News, 80, 31. #17594

  11. Arai,N., Kim,T.W., Kubota,H., Matsumoto,Y., & Koinuma,H. (2002) Combinatorial molecular layer epitaxy of Hf based phosphor oxides. Materials Research Society Symposium Proceedings, 700, 31-36. #17578

  12. Ashley,K., Seghal,A., Amis,E.J., Raghavan,D., & Karim,A. (2002) Combinatorial mapping of polymer film wettability on gradient energy surfaces. Materials Research Society Symposium Proceedings, 700, 151-156. #17576

  13. Baeck,S.H., Jaramillo,T.F., Braendli,C., & McFarland,E.W. (2002) Combinatorial Electrochemical Synthesis and Characterization of Tungsten-Based Mixed-Metal Oxides. Journal of Combinatorial Chemistry, 4, 563-568. #17525

  14. Bagley,M. (2002) Combinatorial Strategies in Biology and Chemistry Edited by A. Beck-Sickinger, P. Weber. Synthesis-Stuttgart, 1132. #17602

  15. Bakhtiar,R., Ramos,L., & Tse,F.L.S. (2002) High-throughput mass spectrometric analysis of xenobiotics in biological fluids. Journal of Liquid Chromatography & Related Technologies, 25, 507-540. #17756

  16. Bala,M., Qadar Pasha,M.A., Bhardwaj,D.K., & Pasha,S. (2002) Novel peptidomimics as angiotensin-Converting enzyme inhibitors: A combinatorial approach. Bioorganic & Medicinal Chemistry, 10, 3685-3691. #17527

  17. Ball,K.D., Erman,B., & Dill,K.A. (2002) The elastic net algorithm and protein structure prediction. J. Comput. Chem., 23, 77-83. #17823

  18. Bannwarth,W., Glatz,H.M., Kohl,M., Schwinn,D., & Tzschucke,C.C. (2002) Fluorous phase chemistry: Fundamentals and applications in catalysis. G. I. T. Laboratory Journal, Europe, 6, 23-24. #17739

  19. Barrett,A.G.M., Hopkins,B.T., & Koebberling,J. (2002) ROMPgel Reagents in Parallel Synthesis. Chemical Reviews (Washington, DC, United States), 102, 3301-3323. #17524

  20. Baruah,M., & Bols,M. (2002) Substitution of .alpha.-azido ethers with Grignard reagents and its use in combinatorial chemistry. Journal of the Chemical Society, Perkin Transactions 1, 509-512. #17788

  21. Batra,S., Srinivasan,T., Rastogi,S.K., & Kundu,B. (2002) Identification of enzyme inhibitors using combinatorial libraries. Curr. Med. Chem., 9, 307-319. #17733

  22. Batra,S., Srinivasan,T., Rastogi,S.K., Kundu,B., Patra,A., Bhaduri,A.P., & Dixit,M. (2002) Corrigendum to \"Combinatorial Synthesis and Biological Evaluation of Isoxazole-Based Libraries as Antithrombotic Agents\" [Bioorg. Med. Chem. Lett. 12 (2002) 1905]. Bioorganic & Medicinal Chemistry Letters, 12, 3349. #17485

  23. Bauser,M. (2002) Preparative high-performance liquid chromatography-mass spectrometry for the high-throughput purification of combinatorial libraries. J. Chromatogr. Sci., 40, 292-296. #17642

  24. Baxendale,I.R., Ley,S.V., & Sneddon,H.F. (2002) A clean conversion of aldehydes to nitriles using a solid-supported hydrazine. Synlett, 775-777. #17695

  25. Belosludov,R.V., Sakahara,S., Yajima,K., Takami,S., Kubo,M., & Miyamoto,A. (2002) Combinatorial computational chemistry approach as a promising method for design of Fischer-Tropsch catalysts based on Fe and Co. Applied Surface Science, 189, 245-252. #17622

  26. Bendale,P.M., & Sun,C.M. (2002) Rapid Microwave-Assisted Liquid-Phase Combinatorial Synthesis of 2-(Arylamino)benzimidazoles. Journal of Combinatorial Chemistry, 4, 359-361. #17694

  27. Beresford,A.P., Selick,H.E., & Tarbit,M.H. (2002) The emerging importance of predictive ADME simulation in drug discovery. Drug Disc. Today, 7, 109-116. #17814

  28. Berg,T., Cohen,S.B., Desharnais,J., Sonderegger,C., Maslyar,D.J., Goldberg,J., Boger,D.L., & Vogt,P.K. (2002) Small-molecule antagonists of Myc/max dimerization inhibit Myc-induced transformation of chicken embryo fibroblasts. Proc. Natl. Acad. Sci. USA, 99, 3830-3835. #17735

  29. Bergmeier,S.C., & Katz,S.J. (2002) A Method for the Parallel Synthesis of Multiply Substituted Oxazolidinones. Journal of Combinatorial Chemistry, 4, 162-166. #17806

  30. Blaney,P., Grigg,R., & Sridharan,V. (2002) Traceless Solid-Phase Organic Synthesis. Chemical Reviews (Washington, DC, United States), 102, 2607-2624. #17650

  31. Blatt,N.B., Bednarski,J.J., Warner,R.E., Leonetti,F., Johnson,K.M., Boitano,A., Yung,R., Richardson,B.C., Johnson,K.J., Ellman,J.A., Opipari,A.W., Jr., & Glick,G.D. (2002) Benzodiazepine-induced superoxide signals B cell apoptosis: mechanistic insight and potential therapeutic utility. J. Clin. Invest., 110, 1123-1132. #17484

  32. Blodgett,J., Wang,Y., Li,T., Polavarapu,P.L., Drabowicz,J., Pietrusiewicz,K.M., & Zygo,K. (2002) Resolution of tert-butyl-1-(2-methylnaphthyl)phosphine oxide using selectors identified from a chemical combinatorial library. Anal. Chem., 74, 5212-5216. #17518

  33. Botta,M., Corelli,F., Petricci,E., & Seri,C. (2002) New solid-supported reagents (SSRs) for selective acylation of amines. Heterocycles, 56, 369-377. #17803

  34. Boyle,N.A., & Janda,K.D. (2002) Formats for combinatorial synthesis: solid-phase, liquid-phase and surface. Curr. Opin. Chem. Biol., 6, 339-346. #17660

  35. Brase,S., Gil,C., & Knepper,K. (2002) The recent impact of solid-phase synthesis on medicinally relevant benzannelated nitrogen heterocycles. Bioorganic & Medicinal Chemistry, 10, 2415-2437. #17644

  36. Breinbauer,R., Vetter,I.R., & Waldmann,H. (2002) From protein domains to drug candidates natural products as guiding principles in the design and synthesis of compound libraries. Angewandte Chemie, International Edition, 41, 2878-2890. #17526

  37. Breinbauer,R., Gonthier,E., & Waldmann,H. (2002) Handbook of Combinatorial Chemistry. Edited by Kyriacos C. Nicolaou. R. Hanko and W. Hartwig. Angewandte Chemie, International Edition, 41, 4145-4146. #17448

  38. Briehn,C.A., & Baeuerle,P. (2002) Design and Synthesis of a 256-Membered .pi.-Conjugated Oligomer Library of Regioregular Head-to-Tail Coupled Quater(3-arylthiophene)s. Journal of Combinatorial Chemistry, 4, 457-469. #17583

  39. Briehn,C.A., & Baeuerle,P. (2002) From solid-phase synthesis of .pi.-conjugated oligomers to combinatorial library construction and screening. Chemical Communications (Cambridge, United Kingdom), 1015-1023. #18006

  40. Broo,K., Larsson,A.K., Jemth,P., & Mannervik,B. (2002) An ensemble of Theta class glutathione transferases with novel catalytic properties generated by stochastic recombination of fragments of two mammalian enzymes. J. Mol. Biol., 318, 59-70. #17646

  41. Bruckdorfer,T. (2002) Parallel synthesis with reactive gases at pressures to 100 bar. GIT Labor-Fachzeitschrift, 46, 505-508. #17636

  42. Brueggemeier,R.W., Richards,J.A., Joomprabutra,S., Bhat,A.S., & Whetstone,J.L. (2002) Molecular pharmacology of aromatase and its regulation by endogenous and exogenous agents. Journal of Steroid Biochemistry and Molecular Biology, 79, 75-84. #17790

  43. Brun,V., Legraverend,M., & Grierson,D.S. (2002) Traceless solid-phase synthesis of 2,6,9-trisubstituted purines from resin bound 6-thiopurines. Tetrahedron, 58, 7911-7923. #17515

  44. Bryant,D., Smythe,M., & Tran,T.T. (2002) A subset-orientated algorithm for minimazing the number of steps required for synthesis of cyclic-peptide libraries. Comput. Chem., 26, 113-117. #17446

  45. Burello,E., Bologa,C., Frecer,V., & Miertus,S. (2002) Application of computer assisted combinatorial chemistry in antivirial, antimalarial and anticancer agents design. Molecular Physics, 100, 3187-3198. #17499

  46. Cacabelos,R. (2002) Pharmacogenomics for the treatment of dementia. Annals of Medicine (Stockholm, Sweden), 34, 357-379. #17460

  47. Cacabelos,R. (2002) Pharmacogenomics in Alzheimer's disease. Mini-Reviews in Medicinal Chemistry, 2, 59-84. #17764

  48. Cawse,J.N., & Wroczynski,R.J. (2002) Screening using high dimensional gradient arrays. Preprints - American Chemical Society, Division of Petroleum Chemistry, 47, 259-261. #17522

  49. Chakraborty,T.K., Ghosh,S., & Jayaprakash,S. (2002) Sugar amino acids and their uses in designing bioactive molecules. Curr. Med. Chem., 9, 421-435. #17734

  50. Chakraborty,T.K., Jayaprakash,S., & Ghosh,S. (2002) Sugar amino acid based scaffolds - novel peptidomimetics and their potential in combinatorial synthesis. Comb. Chem. High Throughput Screening, 5, 373-387. #17550

  51. Chao,E.Y., Minick,D.J., Sternbach,D.D., Shearer,B.G., & Collins,J.L. (2002) A Novel Method for the Generation of Nitrile Oxides on a Solid Phase: Application to the Synthesis of Substituted Benzopyranoisoxazoles. Organic Letters, 4, 323-326. #17819

  52. Chauhan,P.M.S., & Kumar,A. (2002) Solid phase synthesis of structurally diverse tetra substituted pyrimidines for potential use in combinatorial chemistry. Comb. Chem. High Throughput Screening, 5, 93-95. #17766

  53. Cheng,A., Diller,D.J., Dixon,S.L., Egan,W.J., Lauri,G., & Merz,K.M., Jr. (2002) Computation of the physico-chemical properties and data mining of large molecular collections. J. Comput. Chem., 23, 172-183. #17822

  54. Cheng,X., & Hochlowski,J. (2002) Current Application of Mass Spectrometry to Combinatorial Chemistry. Anal. Chem., 74, 2679-2690. #17707

  55. Chikyow,T., Ahmet,P., Nakajima,K., Koida,T., Takakura,M., Yoshimoto,M., & Koinuma,H. (2002) A combinatorial approach in oxide/semiconductor interface research for future electronic devices. Applied Surface Science, 189, 284-291. #17619

  56. Chisholm,B., Potyrailo,R., Cawse,J., Brennan,M., Molaison,C., Shaffer,R., Whisenhunt,D., & Olson,D. (2002) Combinatorial chemistry methods for coating development III. An illustration of an experiment conducted with the combinatorial factory. Proceedings of the International Waterborne, High-Solids, and Powder Coatings Symposium, 29th, 125-137. #17537

  57. Chisholm,B., Potyrailo,R., Cawse,J., Shaffer,R., Brennan,M., Molaison,C., Whisenhunt,D., Flanagan,B., Olson,D., Akhave,J., Saunders,D., Mehrabi,A., & Licon,M. (2002) The development of combinatorial chemistry methods for coating development I. Overview of the experimental factory. Progress in Organic Coatings, 45, 313-321. #17497

  58. Chretien,J.R. (2002) The state of the art for chemometrics in analytical chemistry. Analytical and Bioanalytical Chemistry, 372, 511-512. #17727

  59. Coleman,C.M., MacElroy,J.M.D., Gallagher,J.F., & O'Shea,D.F. (2002) Microwave parallel library generation: comparison of a conventional- and microwave-generated substituted 4(5)-sulfanyl-1H-imidazole library. Journal of Combinatorial Chemistry, 4, 87-93. #17835

  60. Congreve,M.S., Ley,S.V., & Scicinski,J.J. (2002) Analytical construct resins for analysis of solid-phase chemistry. Chemistry--A European Journal, 8, 1768-1776. #17708

  61. Conza,M., & Wennemers,H. (2002) Selective Binding of Two-Armed Diketopiperazine Receptors to Side-Chain-Protected Peptides. J. Org. Chem., 67, 2696-2698. #17763

  62. Cork,D., & Hird,N. (2002) Work-up strategies for high-throughput solution synthesis. Drug Disc. Today, 7, 56-63. #17817

  63. Coulon,E., Pinson,J., Bourzat,J.D., Commercon,A., & Pulicani,J.P. (2002) Surface-Modified Carbon Felts: Possible Supports for Combinatorial Chemistry. J. Org. Chem., 67, 8513-8518. #17477

  64. Cournoyer,J.J., Kshirsagar,T., Fantauzzi,P.P., Figliozzi,G.M., Makdessian,T., & Yan,B. (2002) Color test for the detection of resin-bound aldehyde in solid-phase combinatorial synthesis. Journal of Combinatorial Chemistry, 4, 120-124. #17795

  65. Cox,J. (2002) Chemistry encrypted. Chem. Brit., 38, 36-38. #17560

  66. Cox,K.A., White,R.E., & Korfmacher,W.A. (2002) Rapid determination of pharmacokinetic properties of new chemical entities: In vivo approaches. Comb. Chem. High Throughput Screening, 5, 29-37. #17768

  67. Cremer,R., & Neuschutz,D. (2002) Development of functional materials by a composition spread approach. Materials Research Society Symposium Proceedings, 700, 75-84. #17577

  68. Cremer,R., & Richter,S. (2002) Rapid chemical and structural characterization of metastable thin-film libraries by a combination of electron probe microanalysis and scanning x-ray diffraction. Surface and Interface Analysis, 34, 686-689. #17517

  69. Cuccia,L. (2002) Generation of neuraminidase inhibitors via dynamic combinatorial chemistry. Trends Biochem. Sci., 27, 277-278. #17609

  70. Cui,A., Singh,A., & Kaplan,D.L. (2002) Enzyme-Based Molecular Imprinting with Metals. Biomacromolecules, 3, 1353-1358. #17539

  71. Curran,D.P., & Furukawa,T. (2002) Simultaneous Preparation of Four Truncated Analogues of Discodermolide by Fluorous Mixture Synthesis. Organic Letters, 4, 2233-2235. #17654

  72. Curtis,M.A., Opoku,J.A., Rangarajan,M., Gallagher,A., Sterne,J.A.C., Reid,C.R., Evans,H.E.A., & Samuelsson,B. (2002) Attenuation of the virulence of Porphyromonas gingivalis by using a specific synthetic Kgp protease inhibitor. Infec. Immunity, 70, 6968-6975. #17450

  73. De Mello,A.J. (2002) Miniaturization. Analytical and Bioanalytical Chemistry, 372, 12-13. #17730

  74. Dehli,J.R., & Gotor,V. (2002) Parallel kinetic resolution of racemic mixtures: a new strategy for the preparation of enantiopure compounds? Chem. Soc. Rev., 31, 365-370. #17480

  75. Demuth,D., Finger,K.E., Hill,J.R., Levine,S.M., Lowenhauser,G., Newsam,J.M., Strehlau,W., Tucker,J., & Vietze,U. (2002) Developing combinatorial support for high-throughput experimentation applied to heterogeneous catalysis. ACS Symposium Series, 814, 147-164. #17528

  76. Derouane,E.G. (2002) Challenges and strategies for the implementation of combinatorial methods and high throughput testing in heterogeneous catalysis. NATO Science Series, II: Mathematics, Physics and Chemistry, 69, 3-12. #17458

  77. Ding,S., Gray,N.S., Wu,X., Ding,Q., & Schultz,P.G. (2002) A Combinatorial Scaffold Approach toward Kinase-Directed Heterocycle Libraries. J. Amer. Chem. Soc., 124, 1594-1596. #17797

  78. Doi, Hirofumi Bioinformatics and genomic drug discovery. In: Anonymous. (Eds.) Genomu Soyaku no Saizensen. #17783NEW

  79. Dokoutchaev,A.G., Abdelrazzaq,F., Thompson,M.E., Willson,J., Chang,C., & Bocarsly,A. (2002) Multicomponent Electrodes for Water Oxidation: From Combinatorial to Individual Electrode Study. Chemistry of Materials, 14, 3343-3348. #17603

  80. Durham,T.B., & Miller,M.J. (2002) Conversion of Glucuronic Acid Glycosides to Novel Bicyclic .beta.-Lactams. Organic Letters, 4, 135-138. #17830

  81. Edwards,P.J. (2002) Moving beyond combinatorial chemistry for greater efficiency in lead discovery. JALA, 7, 59-63. #17759

  82. Eksterowicz,J.E., Evensen,E., Lemmen,C., Patrick Brady,G., Kevin Lanctot,J., Bradley,E.K., Saiah,E., Robinson,L.A., Grootenhuis,P.D.J., & Blaney,J.M. (2002) Coupling structure-based design with combinatorial chemistry: application of active site derived pharmacophores with informative library design. Journal of Molecular Graphics & Modelling, 20, 469-477. #17729

  83. Erhardt,P.W. (2002) Medicinal chemistry in the new millennium. A glance into the future. Pure Appl. Chem., 74, 703-785. #17585

  84. Evans,C.A., & Miller,S.J. (2002) Proton-activated fluorescence as a tool for simultaneous screening of combinatorial chemical reactions. Curr. Opin. Chem. Biol., 6, 333-338. #17661

  85. Fang,L., Demee,M., Sierra,T., Kshirsagar,T., Celebi,A.A., & Yan,B. (2002) Kinetics Study of Amine Cleavage Reactions of Various Resin-Bound Thiophenol Esters from Marshall Linker. Journal of Combinatorial Chemistry, 4, 362-368. #17655

  86. Felix,A.M. (2002) Solid-phase peptide synthesis: Bruce Merrifield. Kobunshi, 51, 630-632. #17542

  87. Fernandez,E., Garcia-Ochoa,S., Huss,S., Mallo,A., Bueno,J.M., Micheli,F., Paio,A., Piga,E., & Zarantonello,P. (2002) Solid-phase versus solution synthesis of asymmetrically disubstituted furazano[3,4-b]pyrazines. Tetrahedron Lett., 43, 4741-4745. #17610

  88. Fontaine,L., Lemele,T., Brosse,J.C., Sennyey,G., Senet,J.P., & Wattiez,D. (2002) Grafting of 2-vinyl-4,4-dimethylazlactone onto electron-beam activated poly(propylene) films and fabrics. Application to the immobilization of sericin. Macromolecular Chemistry and Physics, 203, 1377-1384. #17544

  89. Fraga-Dubreuil,J., Famelart,M.H., & Bazureau,J.P. (2002) Ecofriendly Fast Synthesis of Hydrophilic Poly(ethyleneglycol)-Ionic Liquid Matrices for Liquid-Phase Organic Synthesis. Organic Process Research & Development, 6, 374-378. #17653

  90. Fried,H.U., Fuss,S.H., & Korsching,S.I. (2002) Selective imaging of presynaptic activity in the mouse olfactory bulb shows concentration and structure dependence of odor responses in identified glomeruli. Proc. Natl. Acad. Sci. USA, 99, 3222-3227. #17757

  91. Fujii,I. (2002) Development of phage display. High activation of catalytic antibodies. Kagaku to Seibutsu, 40, 396-401. #17604

  92. Fujita,S. (2002) The unit-subduced-cycle-index methods and the characteristic-monomial method. Their relationship as group-theoretical tools for chemical combinatorics. J. Math. Chem., 30, 249-270. #17611

  93. Fukase,K. (2002) Combinatorial synthesis: Solution-phase synthesis and solid-phase split and mixed synthesis. J. Syn. Org. Chem. Jpn., 60, 442-453. #17684

  94. Fukase,K. (2002) Combinatorial chemistry: approach from organic chemistry. Kagaku Furontia, 5, 192-199. #17564

  95. Gallagher,J.F., Coleman,C.M., & O'Shea,D.F. (2002) Ethyl 2-{[2-(3-nitrophenyl)-5-phenyl-1H-imidazol-4-yl]sulfanyl}acetate: synthesis via a microwave-mediated combinatorial chemistry approach. Acta Crystallographica, Section C: Crystal Structure Communications, C58, o139-o141. #17780

  96. Ganesan,A. (2002) Recent developments in combinatorial organic synthesis. Drug Disc. Today, 7, 47-55. #17818

  97. Gangal,R. (2002) DivCalc: A utility for diversity analysis and compound sampling. Molecules [online computer file], 7, 657-661. #17482

  98. Gao,F., Johnson,D.L., Ekins,S., Janiszewski,J., Kelly,K.G., Meyer,R.D., & West,M. (2002) Optimizing higher throughput methods to assess drug-drug interactions for CYP1A2, CYP2C9, CYP2C19, CYP2D6, rCYP2D6, and CYP3A4 in vitro using a single point IC50. J. Biomol. Screen., 7, 373-382. #17502

  99. Garcia-Anton,J.M., Carreno,C., Bonilla,A., & Parente,A. (2002) Combinatorial chemistry: Potential applications as a new lead discovery tool. Comunicaciones presentadas a la Jornadas del Comite Espanol de la Detergencia, 32, 165-174. #17668

  100. Ge,N., Cho,S.J., Hermsmeier,M., Poss,M., & Shen,C.F. (2002) Testing non-additivity of biological activity in a combinatorial library. Comb. Chem. High Throughput Screening, 5, 147-154. #17713

  101. Gebbink,R.J.M.K., Kruithof,C.A., Van Klink,G.P.M., & Van Koten,G. (2002) Dendritic supports in organic synthesis. Reviews in Molecular Biotechnology, 90, 183-193. #17741

  102. Gedey,S., Van der Eycken,J., & Fueloep,F. (2002) Liquid-Phase Combinatorial Synthesis of Alicyclic .beta.-Lactams via Ugi Four-Component Reaction. Organic Letters, 4, 1967-1969. #17703

  103. Godden,J.W., Xue,L., Kitchen,D.B., Stahura,F.L., Schermerhorn,E.J., & Bajorath,J. (2002) Median partitioning: A novel method for the selection of representative subsets from large compound pools. Journal of Chemical Information and Computer Sciences, 42, 885-893. #17630

  104. Goldman,I.D. (2002) Membrane transport of chemotherapeutics and drug resistance: Beyond the ABC family of exporters to the role of carrier-mediated processes. Clinical Cancer Research, 8, 4-6. #17784

  105. Gooding,O.W., Vo,L., Bhattacharyya,S., & Labadie,J.W. (2002) Use of Statistical Design of Experiments in the Optimization of Amide Synthesis Utilizing Polystyrene-Supported N-Hydroxybenzotriazole Resin. Journal of Combinatorial Chemistry, 4, 576-583. #17543

  106. Gravel,M., Thompson,K.A., Zak,M., Berube,C., & Hall,D.G. (2002) Universal Solid-Phase Approach for the Immobilization, Derivatization, and Resin-to-Resin Transfer Reactions of Boronic Acids. J. Org. Chem., 67, 3-15. #17836

  107. Greenbaum,D., Baruch,A., Hayrapetian,L., Darula,Z., Burlingame,A., Medzihradszky,K.F., & Bogyo,M. (2002) Chemical approaches for functionally probing the proteome. Molecular and Cellular Proteomics, 1, 60-68. #17785

  108. Greene,N. (2002) Computer systems for the prediction of toxicity: an update. Advan. Drug Delivery Rev., 54, 417-431. #17749

  109. Gronwald,O., Snip,E., & Shinkai,S. (2002) Gelators for organic liquids based on self-assembly: a new facet of supramolecular and combinatorial chemistry. Current Opinion in Colloid & Interface Science, 7, 148-156. #17687

  110. Grosshans,I., Karl,H., & Stritzker,B. (2002) Combinatorial synthesis of ZnTe nanocrystals in SiO2 on silicon by ion implantation. Nuclear Instruments & Methods in Physics Research, Section B: Beam Interactions with Materials and Atoms, 190, 865-868. #17706

  111. Grzybowski,B.A., Ishchenko,A.V., Shimada,J., & Shakhnovich,E.I. (2002) From Knowledge-Based Potentials to Combinatorial Lead Design in Silico. Account. Chem. Res., 35, 261-269. #17717

  112. Guessregen,S., Wendt,B., & Warne,M. (2002) Approaches to library design for combinatorial chemistry. Methods in Molecular Biology (Totowa, NJ, United States), 201, 277-295. #17507

  113. Gutierrez-de-Teran,H., Lozano,J.J., Segarra,V., & Sanz,F. (2002) Molecular diversity sample generation on the basis of quantum-mechanical computations and principal component analysis. Comb. Chem. High Throughput Screening, 5, 49-57. #17767

  114. Hagemeyer,A., Borade,R., Desrosiers,P., Guan,S., Lowe,D.M., Poojary,D.M., Turner,H., Weinberg,H., Zhou,X., Armbrust,R., Fengler,G., & Notheis,U. (2002) Application of combinatorial catalysis for the direct amination of benzene to aniline. Applied Catalysis, A: General, 227, 43-61. #17787

  115. Hansen,P.R. (2002) Modern chemistry. Peptides and peptide libraries. Dansk Kemi, 83, 25-28. #18008

  116. Harmon,L.A., Schlosser,S.G., & Vayda,A.J. (2002) The role of informatics in combinatorial materials discovery. ACS Symposium Series, 814, 129-145. #17529

  117. Haschke,M., Klein,J., Stichert,W., & Vietze,U. (2002) High throughput experimentation (HTE) with .mu.-X-ray fluorescence. GIT Labor-Fachzeitschrift, 46, 780-782. #17546

  118. Hatanaka,Y., & Sadakane,Y. (2002) Photoaffinity labeling in drug discovery and developments: chemical gateway for entering proteomic frontier. Current Topics in Medicinal Chemistry (Hilversum, Netherlands), 2, 271-288. #17731

  119. He,G., Iijima,T., & Funakubo,H. (2002) New preparation process of Pb(ZrxTi1-x)O3 thin films from PbZrO3 and PbTiO3 multilayers. Journal of Materials Research, 17, 2217-2226. #17514

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  371. Wolf,C., & Hawes,P.A. (2002) A High-Throughput Screening Protocol for Fast Evaluation of Enantioselective Catalysts. J. Org. Chem., 67, 2727-2729. #17772

  372. Wu,Z., & Xu,X. (2002) Using affinity selection to screen new drugs in combinatorial libraries. Fenxi Huaxue, 30, 101-106. #17794

  373. Xie,Y., Men,L.j., Yuan,L.w., Wang,L., & Bai,J.l. (2002) Multi-channel fiber-scanning and data acquisition system. Jisuanji Yu Yingyong Huaxue, 19, 129-131. #17595

  374. Xu,J., & Ma,Y. (2002) Solution-phase combinatorial chemistry. Huaxue Tongbao, 65, 145-152. #17641

  375. Xu,J., Zhang,Q., & Wang,X. (2002) Construction of a novel small library of demulsifier polyether by combinatorial chemical method. Huaxue Tongbao, 65, w040-1-w040/4. #17640

  376. Yadav-Bhatnagar,N., Desjonqueres,N., & Mauger,J. (2002) Polymer-supported approach for solution-phase synthesis of cysteine trap protease inhibitors: procedure for straightforward optimization of the P1-P1' pocket. Journal of Combinatorial Chemistry, 4, 49-55. #17832

  377. Yan,B. (2002) Single-bead analysis in combinatorial chemistry. Curr. Opin. Chem. Biol., 6, 328-332. #17662

  378. Yanase,I., Ohtaki,T., & Watanabe,M. (2002) Combinatorial study for ceramics powder by X-ray diffraction. Solid State Ionics, 154-155, 419-424. #17447

  379. Yanase,I., Ohtaki,T., & Watanabe,M. (2002) Combinatorial study on nano-particle mixture prepared by robot system. Applied Surface Science, 189, 292-299. #17618

  380. Yanase,I., Fujimoto,K., Takada,K., Ohtaki,T., & Watanabe,M. (2002) Development of robot system and X-ray powder diffraction for combinatorial materials research. Materials Research Society Symposium Proceedings, 700, 159-165. #17575

  381. Yang,K., Lou,B., & Saneii,H. (2002) Rapid assembly of 2-aminoimidazolones on solid support. Tetrahedron Lett., 43, 4463-4466. #17632

  382. Yang,Z., Zhang,Z., Meanwell,N.A., Kadow,J.F., & Wang,T. (2002) A Strategy for the Synthesis of Aryl .alpha.-Ketoamides Based upon the Acylation of Anions Derived from Cyanomethylamines Followed by Oxidative Cleavage. Organic Letters, 4, 1103-1105. #17774

  383. Yoshida,J.I., & Suga,S. (2002) Basic concepts of \"cation pool\" and \"cation flow\" methods and their applications in conventional and combinatorial organic synthesis. Chemistry--A European Journal, 8, 2650-2658. #17593

  384. Yoshida,J., & Suga,S. (2002) Serial combinatorial synthesis using cation flow method. J. Syn. Org. Chem. Jpn., 60, 482-483. #17679

  385. Yu,J., Zhao,Y., Holterman,M., & Venton,D.L. (2002) Cocaine detoxification by combinatorially substituted .beta.-Cyclodextrin libraries. Bioorganic & Medicinal Chemistry, 10, 3291-3299. #17566

  386. Yu,Z., & Bradley,M. (2002) Solid supports for combinatorial chemistry. Curr. Opin. Chem. Biol., 6, 347-352. #17659

  387. Yurek,D.A., Branch,D.L., & Kuo,M.S. (2002) Development of a system to evaluate compound identity, purity, and concentration in a single experiment and its application in quality assessment of combinatorial libraries and screening hits. Journal of Combinatorial Chemistry, 4, 138-148. #17798

  388. Zahradnik,R. (2002) Chemistry 2002. Chemicke Listy, 96, 725-737. #17476

  389. Zech,T. (2002) Miniaturized screening system for heterogeneous combinatorial catalysts. Fortschritt-Berichte VDI, Reihe 3: Verfahrenstechnik, 732, i-ix,1. #17592

  390. Zeon,I.W., Sohn,K.S., Park,H.D., & Ryu,S.K. (2002) Synthesis and luminescent properties analysis of Y(As, Nb, P, V)O4 blue emitting phosphors by combinatorial chemistry method. Hwahak Konghak, 40, 63-69. #17701

  391. Zeon,W., Sohn,K.S., & Park,H.D. (2002) Synthesis and photoluminescence properties of Y1-x(P1-y-zNbyVz)O4:Eux phosphors by modified combinatorial chemistry method. Journal of the Korean Chemical Society, 46, 69-75. #17771

  392. Zhang,H., Hoogenboom,R., Fijten,M.W.M., & Schubert,U.S. (2002) Screening and application of ATRP catalysts utilizing an automated synthesizer. Polymer Preprints (American Chemical Society, Division of Polymer Chemistry), 43, 17. #17547

  393. Zhang,S.D., Liu,G., Xia,S.Q., Wu,P., & Zhang,L. (2002) \"Meshed-Bag Gathered-Bunch\" Method for Solid-Phase Synthesis of Small Molecular Diverse Compounds. Journal of Combinatorial Chemistry, 4, 131-137. #17802

  394. Zhang,W., Luo,Z., Chen,C.H.-T., & Curran,D.P. (2002) Solution-Phase Preparation of a 560-Compound Library of Individual Pure Mappicine Analogues by Fluorous Mixture Synthesis. J. Amer. Chem. Soc., 124, 10443-10450. #17563

  395. Zhang,Y., & Amzel,L.M. (2002) Tuberculosis drug targets. Current Drug Targets, 3, 131-154. #17722

  396. Zheng,X.F.S., & Chan,T.F. (2002) Chemical genomics: a systematic approach in biological research and drug discovery. Current Issues in Molecular Biology, 4, 33-43. #17718

  397. Zhu,Q., Yoon,H.S., Parikh,P.B., Chang,Y.T., & Yao,S.Q. (2002) Combinatorial discovery of novel fluorescent dyes based on Dapoxyl. Tetrahedron Lett., 43, 5083-5086. #17600

Thursday, December 12, 2002