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Papers on solid phase organic synthesis published in 1995

This list is arranged by the name of the first author. Any omissions, mistakes and inconsistencies please communicate to the authors of compilation (michal@5z.com). (If you are pointing to any reference, please use its ID# -- the last number in the reference.) You are welcome to use this compilation in your work. Proper way to quote it in your paper is: Lebl M., Leblova Z.: Dynamic database of references in molecular diversity. Internet http://www.5z.com.

Recently added entries are marked in bold

  1. Adamczyk, M., Fishpaugh, J.R., & Mattingly, P.G. (1995) An easy preparation of hapten active esters via solid supported EDAC. Tetrahedron Lett., 36, 8345-8346. #3386

  2. Anderson, R.C., Stokes, J.P., & Shapiro, M.J. (1995) Structure determination in combinatorial chemistry: Utilization of magic angle spinning HMQC and TOCSY NMR spectra in the structure determination of Wang-bound lysine. Tetrahedron Lett., 36, 5311-5314. #2827

  3. Anderson, R. C., Jarema, M. A., Shapiro, M. J., Stokes, J. P., and Ziliox, M. NMR techniques in combinatorial chemistry. 1995. #12543

  4. Aurell, M.J., Boix, C., Ceita, M.L., Llopis, C., Tortajada, A., & Mestres, R. (1995) Polymer supported o-nitrophenylethylene glycols for photoremovable protection of aldehydes. J. Chem. Res-M, 35, 2569-2583. #5605

  5. Auzanneau, F.I., Meldal, M., & Bock, K. (1995) Synthesis, characterization and biocompatibility of PEGA resins. J. Peptide Sci., 1, 31-44. #10795

  6. Baldwin, J.J., Burbaum, J.J., Chelsky, D., Dillard, L.W., Henderson, I., Li, G., Ohlmeyer, M.H.J., Randle, T.L., & Reader, J.C. (1995) Combinatorial libraries encoded with electrophoric tags. Eur. J. Med. Chem., 30 (supplement), 349s-358s. #2807

  7. Baldwin, J.J., Burbaum, J.J., Henderson, I., & Ohlmeyer, M.H.J. (1995) Synthesis of a small molecule combinatorial library encoded with molecular tags. J. Amer. Chem. Soc., 117, 5588-5589. #2737

  8. Bao, Z.N., Chan, W.K., & Yu, L.P. (1995) Exploration of the Stille coupling reaction for the syntheses of functional polymers. J. Amer. Chem. Soc., 117, 12426-12426. #5559

  9. Basu, S., & Wickstrom, E. (1995) Solid phase synthesis of a D-peptide-phosphorothioate oligodeoxynucleotide conjugate from two arms of a polyethylene glycol-polystyrene support. Tetrahedron Lett., 36, 4943-4946. #3044

  10. Beebe, X., Chiappari, C.L., Olmstead, M.M., Kurth, M.J., & Schore, N.E. (1995) Polymer-supported synthesis of cyclic ethers: Electrophilic cyclization of tetrahydrofuroisoxazolines. J. Org. Chem., 60, 4204-4212. #3490

  11. Beebe, X., Schore, N.E., & Kurth, M.J. (1995) Polymer-supported synthesis of cyclic ethers: Electrophilic cyclization of isoxazolines. J. Org. Chem., 60, 4196-4203. #3477

  12. Bergmann, F., Kueng, E., Iaiza, P., & Bannwarth, W. (1995) Allyl as internucleotide protecting group in DNA synthesis to be cleaved off by ammonia. Tetrahedron, 51, 6971-6976. #5609

  13. Bergmann, F., & Bannwarth, W. (1995) Solid phase synthesis of directly linked peptide-oligodeoxynucleotide hybrids using standard synthesis protocols. Tetrahedron Lett., 36, 1839-1842. #2494

  14. Bergmann, F., Bannwarth, W., & Tam, S. (1995) Solid phase synthesis of directly linked PNA-DNA-hybrids. Tetrahedron Lett., 36, 6823-6826. #3159

  15. Bharathi, P., Patel, U., Kawaguchi, T., Pesak, D.J., & Moore, J.S. (1995) Improvements in the synthesis of phenylacetylene monodendrons including a solid-phase convergent method. Macromolecules, 28, 5955. #14282 NEWOLD

  16. Boehm, T.L., & Showalter, H.D.H. (1995) Expedient method for the solid-phase synthesis of aspartic acid protease inhibitors directed toward the generation of libraries. Chemtracts:Org. Chem., 8, 331-335. #3466

  17. Bomann, M.D., Guch, I.C., & DiMare, M. (1995) A mild, pyridine-borane-based reductive amination protocol. J. Org. Chem., 60, 5995-5996. #3177

  18. Boojamra, C.G., Burow, K.M., & Ellman, J.A. (1995) An expedient and high-yielding method for the solid-phase synthesis of diverse 1,4-benzodiazepine-2,5-diones. J. Org. Chem., 60, 5742-5743. #3174

  19. Bray, A.M., Chiefari, D.S., Valerio, R.M., & Maeji, N.J. (1995) Rapid optimization of organic reactions on solid phase using multipin approach: Synthesis of 4-aminoproline analogues by reductive amination. Tetrahedron Lett., 36, 5081-5084. #2804

  20. Brill, W.K.D. (1995) Thioalkylation of nucleoside-H-phosphonates and its application to solid-phase synthesis of oligonucleotides. Tetrahedron Lett., 36, 703-706. #2694

  21. Brown, B.B., Wagner, D.S., & Geysen, H.M. (1995) A single-bead decode strategy using electrospray ionization mass spectrometry and a new photolabile linker: 3-Amino-3-(2- nitrophenyl)-propionic acid. Mol. Diversity, 1, 4-12. #2821 (Available on Internet)

  22. Burbaum, J.J., Ohlmeyer, M.H.J., Reader, J.C., Henderson, I., Dillard, L.W., Li, G., Randle, T.L., Sigal, N.H., Chelsky, D., & Baldwin, J.J. (1995) A paradigm for drug discovery employing encoded combinatorial libraries. Proc. Natl. Acad. Sci. USA, 92, 6027-6031. #2732

  23. Burger, M.T., & Still, W.C. (1995) Synthetic ionophores. Encoded combinatorial libraries of cyclen- based receptors for Cu(2+) and Co(2+). J. Org. Chem., 60, 7382-7383. #3355

  24. Burgess, K., Linthicum, D.S., & Shin, H. (1995) Solid phase syntheses of unnatural biopolymers containing repeating urea units. Angew. Chem. Int. Ed., 34, 907-909. #3583

  25. Campbell, D.A., Bermak, J.C., Burkoth, T.S., & Patel, D.V. (1995) A transition state analogue inhibitor combinatorial library. J. Amer. Chem. Soc., 117, 5381-5382. #2727

  26. Cao, X., Moran, E.J., Siev, D., Lio, A., Ohashi, C., & Mjalli, A.M.M. (1995) Synthesis of NH-acyl-alpha-aminoamides on Rink resin: Inhibitors of the hematopoietic protein tyrosine phosphatase (HePTP). Bioorg. Med. Chem. Lett., 5, 2953-2958. #10540

  27. Cargill, J. F., Maiefski, R. R., and Toyonaga, B. E. Automated combinatorial chemistry on solid phase. In: Anonymous. (Eds.) Zymark Corporation, Hopkinton, MA p.221 Proceedingds of the 13th International Symposium of Laboratory Robotics and Automation 1995. #8300

  28. Chabala, J.C. (1995) Solid-phase combinatorial chemistry and novel tagging methods for identifying leads. Curr. Opin. Biotechnol., 6, 632-639. #4916

  29. Chabala, J.C., Baldwin, J.J., Burbaum, J.J., Chelsky, D., Dillard, L.W., Henderson, I., Li, G., Ohlmeyer, M.H.J., Randle, T.L., Reader, J.C., Rokosz, L., & Sigal, N.H. (1995) Binary encoded small-molecule libraries in drug discovery and optimization. Perspect. Drug Disc. Design, 2, 305-318. #2905

  30. Chan, W.C., & Mellor, S.L. (1995) Reductive alkylation of 9-amino-xanthen-3-yloxymethylpoly(styrene): A novel procedure for the synthesis of peptidyl N-alkyl amides by Fmoc/But chemistry. J. Chem. Soc. Chem. Commun., 1475-1477. #5618

  31. Chenera, B., Finkelstein, J.A., & Veber, D.F. (1995) Protodetachable arylsilane polymer linkages for use in solid phase organic synthesis. J. Amer. Chem. Soc., 117, 11999-12000. #3375

  32. Chu, S.S., & Reich, S.H. (1995) NPIT: A new reagent for quantitatively monitoring reactions of amines in combinatorial synthesis. Bioorg. Med. Chem. Lett., 5, 1053-1058. #3224

  33. Criton, M., Dewynter, G., Aouf, N., Montero, J.L., & Imbach, J.L. (1995) Nucleopeptidic bioconjugates containing a sulfamide bridge: Linkage via the Mitsunobu reaction. Nucleosides Nucleotides, 14, 1795-1801. #6239

  34. Cuervo, J.H., Weitl, F., Ostresh, J.M., Hamashin, V.T., Hannah, A.L. & Houghten, R.A. (1995) Polyalkylamine chemical combinatorial libraries. In H.L.S. Maia (Ed.), Peptides 94, Proc.23.EPS. (pp. 465-466). ESCOM, Leiden. #2846

  35. Dankwardt, S.M., Newman, S.R., & Krstenansky, J.L. (1995) Solid phase synthesis of aryl and benzylpiperazines and their application in combinatorial chemistry. Tetrahedron Lett., 36, 4923-4926. #2805

  36. Dapremont, L., Valerio, R.M., Bray, A.M., Stewart, K.M., Mason, T.J., Wang, A.W., & Maeji, N.J. (1995) Multiple synthesis using the multipin method. Physiol. Chem. Phys. Med. NMR, 27, 339-343. #5215

  37. Das, S.K., Kumar, A.J., Nandrajog, S., & Kumar, A. (1995) Polymer supported VO(2+) Schiff base catalyst for hydroxylation of benzene. Tetrahedron Lett., 36, 7909-7912. #5627

  38. Deleuze, H., & Sherrington, D.C. (1995) Poly(p-acetoxylstyrene) resin: A prospective new support for combinatorial synthesis. J. Chem. Soc. Perkin Trans. 2, 36, 2217-2221. #5628

  39. Dempcy, R.O., Browne, K.A., & Bruice, T.C. (1995) Synthesis of the polycation thymidyl DNG, its fidelity in binding polyanionic DNA/RNA, and the stability and nature of the hybrid complexes. J. Amer. Chem. Soc., 117, 6140-6141. #14274 NEWOLD

  40. DeSilva, B.S., & Wilson, G.S. (1995) Solid phase synthesis of bifunctional antibodies. J. Immunol. Method, 188, 9-19. #3729

  41. DeWitt, S.H., Schroeder, M.C., & Stankovic, C.J. (1995) Integration and automation of multiple, simultaneous organic synthesis on a solid support. Amer. Lab., 26AA-26BB. #2421

  42. Dumy, P., Eggleston, I.M., Cervigni, S., Sila, U., Sun, X., & Mutter, M. (1995) A convenient synthesis of cyclic peptides as regioselectively addressable functionalized templates (RAFT). Tetrahedron Lett., 36, 1255-1258. #2353

  43. Ecker, D.J., & Crooke, S.T. (1995) Combinatorial drug discovery: Which methods will produce the greatest value? Biotechnology, 13, 351-360. #4056

  44. Egner, B.J., Langley, G.J., & Bradley, M. (1995) Solid phase chemistry: Direct monitoring by matrix-assisted laser desorption/ionization time of flight mass spectrometry.A tool for combinatorial chemistry. J. Org. Chem., 60, 2652-2653. #2639

  45. Fehrentz, J.A., Paris, M., Heitz, A., Velek, J., Liu, C.F., Winternitz, F., & Martinez, J. (1995) Improved solid phase synthesis of C-terminal peptide aldehydes. Tetrahedron Lett., 36, 7871-7874. #3265

  46. Flegelova, Z., Krchnak, V., Sepetov, N.F., Stankova, M., Issakova, O., Cabel, D., Lam, K.S. & Lebl, M. (1995) Libraries of small compact structures based on N-acyl-N- alkylamino acids. In H.L.S. Maia (Ed.), Peptides 94, Proc.23.EPS. (pp. 469-470). ESCOM, Leiden. #1347

  47. Fodor, S.P.A. (1995) Photolithography and biopolymer synthesis. In Anonymous, Book of Abstracts, 210th ACS National Meeting, Chicago, IL, August 20-24. (pp. PMSE-224. American Chemical Society,Washington,D, #6412

  48. Forman, F.W., & Sucholeiki, I. (1995) Solid-phase synthesis of biaryls via the Stille reaction. J. Org. Chem., 60, 523-528. #2304

  49. Franot, C., Stone, G.B., Engeli, P., Spondlin, C., & Waldvogel, E. (1995) A polymer-bound oxazaborolidine catalyst: Enantioselective borane reductions of ketones. Tetrahedron:Asymmetry, 6, 2755-2766. #5636

  50. Gasparrini, F., Misiti, D., & Villani, C. (1995) Enantioselective recognition by a new chiral stationary phase at receptorial level. J. Org. Chem., 60, 4314-4315. #2826

  51. Gennari, C., Nestler, H.P., Salom, B., & Still, W.C. (1995) Solid-phase synthesis of vinylogous sulphonyl peptides. Angew. Chem. Int. Ed., 34, 1763-1765. #3207

  52. Gennari, C., Nestler, H.P., Salom, B., & Still, W.C. (1995) Synthetic receptors based on vinylogous sulfonyl peptides. Angew. Chem. Int. Ed., 34, 1765-1768. #3208

  53. Goebel, M., & Ugi, I. (1995) Beyond peptide and nucleic acid combinatorial libraries: Applying unions of multicomponent reactions towars the generation of carbohydrate combinatorial libraries. Tetrahedron Lett., 36, 6043-6046. #3115

  54. Goff, D.A., & Zuckermann, R.N. (1995) Solid-phase synthesis of defined 1,4-benzodiazepine-2,5-dione mixtures. J. Org. Chem., 60, 5744-5745. #3175

  55. Goff, D.A., & Zuckermann, R.N. (1995) Solid-phase synthesis of highly substituted peptoid 1(2H)-isoquinolinones. J. Org. Chem., 60, 5748-5749. #3173

  56. Gold, L., Polisky, B., Uhlenbeck, O., & Yarus, M. (1995) Diversity of oligonucleotide functions. Annu. Rev. Biochem., 64, 763-797. #3141

  57. Gordon, D.W., & Steele, J. (1995) Reductive alkylation on a solid phase: Synthesis of a piperazinedione combinatorial library. Bioorg. Med. Chem. Lett., 5, 47-50. #2306

  58. Gordon, E.M. (1995) Libraries of non-polymeric organic molecules. Curr. Opin. Biotechnol., 6, 624-631. #6539

  59. Gordon, E.M., Gallop, M.A., Campbell, D., Holmes, C., Bermak, J., Look, G., Murphy, M., Needels, M., Jacobs, J., Sugarman, J., Chinn, J., Fritsch, B.R., & Jones, D. (1995) Combinatorial organic synthesis: Applications to drug discovery. Eur. J. Med. Chem., 30, 337s-348s. #2806

  60. Green, J. (1995) Solid phase synthesis of lavendustin A and analogues. J. Org. Chem., 60, 4287-4290. #3236

  61. Gregorius, K., Mouritsen, S., & Elsner, H.I. (1995) Hydrocoating: A new method for coupling biomolecules to solid phases. J. Immunol. Method, 181, 65-73. #4911

  62. Grotli, M., & Sproat, B.S. (1995) A universal solid-phase synthesis of branched oligoribonucleotides. J. Chem. Soc. Chem. Commun., 495-497. #2378

  63. Hauske, J.R., & Dorff, P. (1995) A solid phase CBZ chloride equivalent. A new matrix specific linker. Tetrahedron Lett., 36, 1589-1592. #2489

  64. Hiroshige, M., Hauske, J.R., & Zhou, P. (1995) Palladium-mediated macrocyclization on solid support and its applications to combinatorial synthesis. J. Amer. Chem. Soc., 117, 11590-11591. #3353

  65. Hiroshige, M., Hauske, J.R., & Zhou, P. (1995) Formation of C-C bond in solid phase synthesis using the Heck reaction. Tetrahedron Lett., 36, 4567-4570. #3238

  66. Holmes, C.P., & Jones, D.G. (1995) Reagents for combinatorial organic synthesis: Development of a new o-nitrobenzyl photolabile linker for solid phase synthesis. J. Org. Chem., 60, 2318-2319. #2157

  67. Holmes, C.P., Chinn, J.P., Look, G.C., Gordon, E.M., & Gallop, M.A. (1995) Strategies for combinatorial organic synthesis: Solution and polymer-supported synthesis of 4-thiazolidinones and 4-metathiazanones derived from amino acids. J. Org. Chem., 60, 7328-7333. #3312

  68. Hutchins, S.M., & Chapman, K.T. (1995) A strategy for urea linked diamine libraries. Tetrahedron Lett., 36, 2583-2586. #2647

  69. Itsuno, S., Watanabe, K., Koizumi, T., & Ito, K. (1995) Asymmetric diels-alder reaction of cyclopentadiene with methacrolein using polymer-supported chiral catalysts. React. Polym., 24, 219-227. #2605

  70. Johnson, C.R., & Zhang, B. (1995) Solid phase synthesis of alkenes using the Horner-Wadsworth-Emmons reaction and monitoring by gel phase (31)P NMR. Tetrahedron Lett., 36, 9253-9256. #4332

  71. Kaljuste, K., & Und n, A. (1995) Solid phase synthesis of 1,2,3,4-tetrahydro-b-carbolines: Implications for combinatorial chemistry. Tetrahedron Lett., 36, 9211-9214. #3445

  72. Kellenberger, C., Hietter, H., & Luu, B. (1995) Regioselective formation of the three disulfide bonds of a 35-residue insect peptide. Peptide Res., 8, 321-327. #6836

  73. Kester, J., Geldern, T.V., Kalvin, D. & Sowin, T. (1995) Solid-phase synthesis of azole endothelin antagonists. In Anonymous, Book of Abstracts, 210th ACS National Meeting, Chicago, IL, August 20-24. (pp. MEDI-36. American Chemical Society,Washington,D, #6847

  74. Kick, E.K., & Ellman, J.A. (1995) Expedient method for the solid-phase synthesis of aspartic acid protease inhibitors directed toward the generation of libraries. J. Med. Chem., 38, 1427-1430. #2668

  75. Krchnak, V., Flegelova, Z., Weichsel, A.S., & Lebl, M. (1995) Polymer-supported Mitsunobu ether formation and its use in combinatorial chemistry. Tetrahedron Lett., 36, 6193-6196. #2426

  76. Krchnak, V., Weichsel, A.S., Cabel, D., & Lebl, M. (1995) Linear presentation of variable side-chain spacing in a highly diverse combinatorial library. Peptide Res., 8, 198-205. #2723

  77. Lelievre, D., Daguet, D., & Brack, A. (1995) On-line solid-phase synthesis of a peptide bi-derivatized with biotin and 4-azido salicylic acid. Tetrahedron Lett., 36, 9317-9320. #7014

  78. Lenzi, A., Reginato, G., Taddei, M., & Trifilieff, E. (1995) Solid phase synthesis of a self complementary (antiparallel) chiral peptidic nucleic acid strand. Tetrahedron Lett., 36, 1717-1718. #2492

  79. Ley, S.V., Mynett, D.M., & Koot, W.J. (1995) Solid phase synthesis of bicyclo[2.2.2]octane derivatives via tandem Michael addition reactions and subsequent reductive amination. Synlett, 1017-1020. #3358

  80. Li, R., Cohen, F.E. & Kenyon, G.L. (1995) A methodology for the solid phase syntheses of alpha,beta- unsaturated ketone combinatorial libraries. In Anonymous, Book of Abstracts, 210th ACS National Meeting, Chicago, IL, August 20-24. (pp. MEDI-227. American Chemical Society,Washington,D, #7032

  81. Liu, G., & Ellman, J.A. (1995) A general solid-phase synthesis strategy for the preparation of 2-pyrrolidinemethanol ligands. J. Org. Chem., 60, 7712-7713. #3382

  82. Look, G.C., Murphy, M.M., Campbell, D.A., & Gallop, M.A. (1995) Trimethylorthoformate: A mild and effective dehydrating reagent for solution and solid phase imine formation. Tetrahedron Lett., 36, 2937-2940. #3043

  83. Martin, E.J., Blaney, J.M., Siani, M.A., Spellmeyer, D.C., Wong, A.K., & Moos, W.H. (1995) Measuring diversity: Experimental design of combinatorial libraries for drug discovery. J. Med. Chem., 38, 1431-1436. #2671

  84. Matson, R.S., Rampal, J.B., Pentoney, S.L.Jr., Anderson, P.D., & Coassin, P. (1995) Biopolymer synthesis on polypropylene supports: Oligonucleotide arrays. Anal. Biochem., 224, 110-116. #10573

  85. Mayer, J.P., Heil, J.R., Zhang, J., & Munson, M.C. (1995) An alternative solid-phase approach ti C(1)-oxytocin. Tetrahedron Lett., 36, 7387-7390. #3263

  86. Meinjohanns, E., Meldal, M., Paulsen, H., & Bock, K. (1995) Dithiasuccinoyl (Dts) amino-protecting group used in syntheses of 1,2-trans-amino sugar glycosides. J. Chem. Soc. Perkin Trans. 1, 405-415. #7165

  87. Meutermans, W.D.F., & Alewood, P.F. (1995) The solid phase synthesis of dihydro- and tetrahydroisoquinolines. Tetrahedron Lett., 36, 7709-7712. #3259

  88. Meyers, H.V., Dilley, G.J., Durgin, T.L., Powers, T.S., Winssinger, N.A., Zhu, H., & Pavia, M.R. (1995) Multiple simultaneous synthesis of phenolic libraries. Mol. Diversity, 1, 13-20. #2823 (Available on Internet)

  89. Mora, N., Lacombe, J.M., & Pavia, A.A. (1995) A new approach to phosphoserine, phosphothreonine and phosphotyrosine synthons and to thiophospho analogs. Stepwise synthesis of mono- and multiphosphorylated phosphopeptides related to src-protein kinase. Int. J. Peptide Prot. Res., 45, 53-63. #7225

  90. Moran, E.J., Sarshar, S., Cargill, J.F., Shahbaz, M.M., Lio, A., Mjalli, A.M.M., & Armstrong, R.W. (1995) Radio frequency tag encoded combinatorial library method for the discovery of tripeptide-substituted cinnamic acid inhibitors of the protein tyrosine phosphatase PTP1B. J. Amer. Chem. Soc., 117, 10787-10788. #3431

  91. Moran, E.J., Wilson, T.E., Cho, C.Y., Cherry, S.R., & Schultz, P.G. (1995) Novel biopolymers for drug discovery. Biopolymers (Pept. Sci. ), 37, 213-219. #2423

  92. Muller, C., Kitas, E., & Wessel, H.P. (1995) Novel oligosaccharide mimetics by solid-phase synthesis. J. Chem. Soc. Chem. Commun., 2425-2426. #5666

  93. Muller, W.T., Klein, D.L., Lee, T., Clarke, J., McEuen, P.L., & Schultz, P.G. (1995) A strategy for the chemical synthesis of nanostructures. Science, 268, 272-273. #3554

  94. Murphy, M.M., Schullek, J.R., Gordon, E.M., & Gallop, M.A. (1995) Combinatorial organic synthesis of highly functionalized pyrrolidines: Identification of a potent angiotensin converting enzyme inhibitor from a mercaptoacyl proline library. J. Amer. Chem. Soc., 117, 7029-7030. #2731

  95. Nguyen, S.T., & Grubbs, R.H. (1995) The synthesis and activities of polystyrene-supported olefin metathesis catalysts based on Cl2(PR3)2Ru=CH-CH=CPh2. J. Organomet. Chem., 497, 195-200. #5667

  96. Ohtani, N., Inoue, Y., Inagaki, Y., Fukuda, K., & Nishiyama, T. (1995) Reactions of amino acid decyl esters with nucleophiles catalyzed by polymer-supported amine-metal complexes. Bull. Chem. Soc. Jpn., 68, 1669-1675. #5668

  97. Otaka, A., Miyoshi, K., Burke, T.R., Roller, P.P., Kubota, H., Tamamura, H., & Fujii, N. (1995) Synthesis and application of N-Boc-L-2-amino-4- (diethylphosphono)-4,4-difluorobutanoic acid for solid-phase synthesis of nonhydrolyzable phosphoserine peptide analogues. Tetrahedron Lett., 36, 927-930. #2700

  98. Patek, M., Drake, B., & Lebl, M. (1995) Solid-phase synthesis of "small" organic molecules based on thiazolidine scaffold. Tetrahedron Lett., 36, 2227-2230. #1356

  99. Peterson, M.L. (1995) Automated strategies for combinatorial chemistry. Biomed. Product, 20, 96-96. #3202

  100. Petrucci, M.G.L., & Kakkar, A.K. (1995) A convenient molecular self-assembly route to thin films containing terminal donor ligands and anchored organotransition- metal complexes for heterogenized homogenous catalysis. J. Chem. Soc. Chem. Commun., 1577-1578. #5669

  101. Peyman, A., Weiser, C., & Uhlmann, E. (1995) Facile preparation of 3'-derivatized oligodeoxynucleotides. Bioorg. Med. Chem. Lett., 5, 2469. #14280 NEWOLD

  102. Plunkett, M.J., & Ellman, J.A. (1995) A silicon-based linker for traceless solid-phase synthesis. J. Org. Chem., 60, 6006-6007. #3307

  103. Plunkett, M.J., & Ellman, J.A. (1995) Solid phase synthesis of structurally diverse 1,4-benzodiazepine derivatives using the Stille coupling reaction. J. Amer. Chem. Soc., 117, 3306-3307. #2159

  104. Randolph, J.T., McClure, K.F., & Danishefsky, S.J. (1995) Major simplifications in oligosaccharide syntheses arising from a solid-phase based method: An application to the synthesis of the Lewis b antigen. J. Amer. Chem. Soc., 117, 5712-5719. #2766

  105. Rano, T.A., & Chapman, K.T. (1995) Solid phase synthesis of aryl ethers via the Mitsunobu reaction. Tetrahedron Lett., 36, 3789-3792. #2725

  106. Richter, L.S., & Zuckermann, R.N. (1995) Synthesis of peptide nucleic acids (PNA) by submonomer solid phase synthesis. Bioorg. Med. Chem. Lett., 5, 1159-1162. #5681

  107. Ruan, F., Yamamura, S., Hakomori, S., & Igarashi, Y. (1995) Synthesis of sphingosine conjugate with controlled pore glass beads. Tetrahedron Lett., 36, 6615-6618. #3162

  108. Rudge, D. and Main, B. Automated chemical synthesis. In: Anonymous. (Eds.) Zymark Corporation, Hopkinton, MA Proceedingds of the International Symposium of Laboratory Robotics and Automation 1994. #8299

  109. Safar, P., Stierandova, A. & Lebl, M. (1995) Amino-acid like subunits based on iminodiacetic acid and their application in linear and DKP libraries. In H.L.S. Maia (Ed.), Peptides 94, Proc.23.EPS. (pp. 471-472). ESCOM, Leiden. #1350

  110. Salmon, S.E., Lam, K.S., Felder, S., Yeoman, H., Schlessinger, J., Ulrich, A., Krchnak, V., & Lebl, M. (1995) Use of large combinatorial chemical libraries for anticancer drug discovery. Int. J. Pharmacogn., 33 Suppl., 67-74. #5254

  111. Sasmor, H.M., Dellinger, D.J., Zenk, P.C., & Lee, L.P. (1995) A practical method for the synthesis and purification of (14)C labeled oligonucleotides. J. Label. Compound. Radiopharm., 36, 15-31. #2705

  112. Seligmann, B., Abdul-Latif, F., Al-Obeidi, F., Flegelova, Z., Issakova, O., Kocis, P., Krchnak, V., Lam, K.S., Lebl, M., Ostrem, J., Safar, P., Sepetov, N., Stierandova, A., Strop, P., & Wildgoose, P. (1995) The construction and use of peptide and non-peptidic combinatorial libraries to discover enzyme inhibitors. Eur. J. Med. Chem., 30 (supplement); Pro, 319s-335s. #2429

  113. Sucholeiki, I. (1995) Solid-phase synthetic methods in combinatorial chemistry. Med. Chem. Res., 5, 618-630. #7807

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